Liu, Minglong; Yoshisada, Ryoji; Amedi, Avand; Hopstaken, Antonius J P; Pascha, Mirte N; de Haan, Cornelis A M; Geerke, Daan P; Poole, David A; Jongkees, Seino A K
(Wiley, 2023-03-07)
Macrocyclisation provides a means of stabilising the conformation of peptides, often resulting in improved stability, selectivity, affinity, and cell permeability. In this work, a new approach to peptide macrocyclisation ...